Combinatorial chemistry and high-throughput screening are indispensable tools used in chemical biology to synthesize diverse chemical libraries and identify potential drug leads. Natural products and their derivatives have historically served as successful drug leads due to their structural complexity and co-evolution within biological systems. Components of natural product scaffolds may serve as beneficial motifs in the development of new biological probes….Continue Reading Synthesis, Biological Screening, and Structure-Activity Relationships of Non-Proteinogenic Cyclic Hexapeptide Libraries